Anticancer Class

Showing 3 drugs starting with: B

Bevacizumab

Brand: Avastin (global) / Bevacizumab (IN/BD)
Class: Anticancer
Subclass: VEGF monoclonal antibody
PK: t½ 480 hours | Clearance: hepatic
Max Dose: 15 day
life-threatening
AE: Hypertension, proteinuria, arterial thromboembolism, GI perforation

Binimetinib

Brand: Mektovi (global)
Class: Anticancer
Subclass: MEK inhibitor
PK: t½ 9 hours | Clearance: hepatic
Max Dose: 90 day
severe
AE: Retinal pigment epithelial detachment, CPK elevations, hepatotoxicity, diarrhea

Brigatinib

Brand: Alunbrig (global)
Class: Anticancer
Subclass: ALK inhibitor (2nd gen)
PK: t½ 26 hours | Clearance: hepatic
Max Dose: 180 day
severe
AE: Pneumonitis (early onset), hypertension, visual disturbances, hyperglycemia, myalgia