Anticancer Class

Showing 5 drugs starting with: D

Dabrafenib

Brand: Tafinlar (global)
Class: Anticancer
Subclass: BRAF inhibitor (V600E/K)
PK: t½ 8 hours | Clearance: hepatic
Max Dose: 300 day
moderate
AE: Fever, hyperglycemia, skin reactions, uveitis

Dasatinib

Brand: Sprycel (US/EU) / Dasatinib (IN/BD)
Class: Anticancer
Subclass: BCR-ABL Tyrosine Kinase Inhibitor
PK: t½ 4 hours | Clearance: hepatic
Max Dose: 140 day
severe
AE: Myelosuppression, pleural effusion, pulmonary hypertension

Daunorubicin

Brand: Cerubidine (global) / Daunoblastin (IN/BD)
Class: Anticancer
Subclass: Anthracycline (topoisomerase II inhibitor)
PK: t½ 19 hours | Clearance: hepatic
Max Dose: not added
life-threatening
AE: Myelosuppression, cardiomyopathy, mucositis, red/orange urine

Docetaxel

Brand: Taxotere (global) / Daxotel (IN/BD)
Class: Anticancer
Subclass: Taxane (microtubule stabilizer)
PK: t½ 11 hours | Clearance: hepatic
Max Dose: not added
severe
AE: Neutropenia, peripheral edema/fluid retention, mucositis, nail changes

Durvalumab

Brand: Imfinzi (global) / Durvalumab (IN/BD)
Class: Anticancer
Subclass: PD-L1 Immune Checkpoint Inhibitor
PK: t½ 432 hours | Clearance: hepatic
Max Dose: 1500 day
life-threatening
AE: Immune pneumonitis, hepatitis, colitis, endocrinopathy