Anticoagulant Class
Showing 3 drugs
starting with: A
Acenocoumarol
Brand: Acitrom / Sintrom / Nicoumalone
Class: Anticoagulant
Subclass: Vitamin K antagonist
PK:
t½ 10 hours | Clearance: hepatic
Max Dose: 6 day
Max Dose: 6 day
severe
AE: Bleeding (GI/intracranial), skin necrosis (rare in protein C/S deficiency), INR variability, teratogenicity
AE: Bleeding (GI/intracranial), skin necrosis (rare in protein C/S deficiency), INR variability, teratogenicity
Apixaban
Brand: Eliquis (US/EU) / Apigat (IN) / Apixava (BD)
Class: Anticoagulant
Subclass: NOAC / DOAC (Xa inhibitor)
PK:
t½ 12 hours | Clearance: mixed
Max Dose: 10 day
Max Dose: 10 day
moderate
AE: Bleeding (especially GI), anemia, rare hypersensitivity
AE: Bleeding (especially GI), anemia, rare hypersensitivity
Argatroban
Brand: Argatroban (US/EU) / Argihope (IN) / Argiprax (IN) / Argatro (BD)
Class: Anticoagulant
Subclass: Direct thrombin inhibitor (parenteral)
PK:
t½ 1 hours | Clearance: hepatic
Max Dose: not added
Max Dose: not added
severe
AE: Bleeding, hypotension, infusion-related reactions, elevated INR during therapy
AE: Bleeding, hypotension, infusion-related reactions, elevated INR during therapy