Antihypertensive Class
Showing 5 drugs
starting with: L
Labetalol
Brand: Trandate (US/EU) / Labeta (IN) / Labocard (BD)
Class: Antihypertensive
Subclass: Combined α₁ + β blocker
PK:
t½ 6 hours | Clearance: hepatic
Max Dose: 1200 day
Max Dose: 1200 day
moderate
AE: Postural hypotension (esp. after IV), fatigue, bradycardia, nasal congestion, scalp tingling
AE: Postural hypotension (esp. after IV), fatigue, bradycardia, nasal congestion, scalp tingling
Lisinopril
Brand: Zestril (US/EU) / Lisoril (IN) / Lisonorm (BD)
Class: Antihypertensive
Subclass: ACE inhibitor (not a prodrug)
PK:
t½ 12 hours | Clearance: renal
Max Dose: 40 day
Max Dose: 40 day
moderate
AE: Dry cough, hyperkalemia, dizziness, hypotension, rare angioedema
AE: Dry cough, hyperkalemia, dizziness, hypotension, rare angioedema
Lisinopril + Hydrochlorothiazide
Brand: Zestoretic
Class: Antihypertensive
Subclass: ACEI + Thiazide diuretic
PK:
t½ 12 hours | Clearance: renal
Max Dose: not added
Max Dose: not added
moderate
AE: Cough, dizziness, hyperkalemia, hyponatremia
AE: Cough, dizziness, hyperkalemia, hyponatremia
Losartan
Brand: Cozaar (US/EU) / Losar (IN) / Losakind (IN) / Lorista (BD)
Class: Antihypertensive
Subclass: Angiotensin II receptor blocker (ARB)
PK:
t½ 9 hours | Clearance: hepatic
Max Dose: 100 day
Max Dose: 100 day
moderate
AE: Dizziness, hyperkalemia (less than ACEIs), renal function changes; rare angioedema
AE: Dizziness, hyperkalemia (less than ACEIs), renal function changes; rare angioedema
Losartan + Hydrochlorothiazide
Brand: Hyzaar
Class: Antihypertensive
Subclass: ARB + Thiazide diuretic
PK:
t½ 6 hours | Clearance: mixed
Max Dose: not added
Max Dose: not added
moderate
AE: Hypotension, dizziness, hyperkalemia, electrolyte imbalance
AE: Hypotension, dizziness, hyperkalemia, electrolyte imbalance