Cardiovascular Class
Pitavastatin
Brand: Livalo (US/EU) / Pivasta (IN) / Pitava (JP)
Subclass: Statin (HMG-CoA reductase inhibitor)
PK:
t½ 12 hours | Clearance: hepatic
Max Dose: 4 day
Max Dose: 4 day
mild
AE: Myalgia, mild liver enzyme elevation
AE: Myalgia, mild liver enzyme elevation
Pravastatin
Brand: Pravachol (US/EU) / Pravator (IN) / Vastatin (BD)
Subclass: Statin (HMG-CoA reductase inhibitor)
PK:
t½ 1.8 hours | Clearance: hepatic
Max Dose: 80 day
Max Dose: 80 day
mild
AE: Mild transaminitis, headache, mild GI upset
AE: Mild transaminitis, headache, mild GI upset
Rosuvastatin
Brand: Crestor (US/EU) / Rosuvas (IN) / Rosumix (BD)
Subclass: Statin (HMG-CoA reductase inhibitor)
PK:
t½ 19 hours | Clearance: hepatic
Max Dose: 40 day
Max Dose: 40 day
moderate
AE: Myalgia, ALT elevation, rare rhabdomyolysis
AE: Myalgia, ALT elevation, rare rhabdomyolysis
Simvastatin
Brand: Zocor (US/EU) / Simvotin (IN) / Simvas (BD)
Subclass: Statin (HMG-CoA reductase inhibitor)
PK:
t½ 2 hours | Clearance: hepatic
Max Dose: 40 day
Max Dose: 40 day
moderate
AE: Myopathy, liver enzyme rise, GI discomfort
AE: Myopathy, liver enzyme rise, GI discomfort